| Sequence | IC50 (nM) |  | Sequence | IC50 (nM) |  | Sequence | IC50 (nM) |
---|---|---|---|---|---|---|---|---|
C366A | AYGVSATKL | 66 | C366K | KYGVSATKL | 15.5 | C366D | DYGVSATKL | 551.5 |
Y367A | CAGVSATKL | 25435 | Y367K | CKGVSATKL | 22549 | Y367 D | CDGVSATKL | 28232 |
G368A | CYAVSATKL | 7.3 | G368K | CYKVSATKL | 18.5 | G368 D | CYDVSATKL | 150 |
V369A | CYGASATKL | 13.8 | V369K | CYGKSATKL | 69.6 | V369 D | CYGDSATKL | 791.1 |
S370A | CYGVAATKL | 216.1 | S370K | CYGVKATKL | 1118 | S370 D | CYGVDATKL | 959.9 |
 | CYGVSATKL | 59.2 | A371K | CYGVSKTKL | 40.3 | A371 D | CYGVSDTKL | 112.9 |
T372A | CYGVSAAKL | 1995 | T372K | CYGVSAKKL | 3122 | T372 D | CYGVSADKL | 882.4 |
K373A | CYGVSATAL | 13.3 | Â | CYGVSATKL | 59.2 | K373 D | CYGVSATDL | 38.5 |
L374A | CYGVSATKA | 9265 | L374K | CYGVSATKK | 22172 | L374 D | CYGVSATKD | 25522 |